Compile Data Set for Download or QSAR
Report error Found 1283 Enz. Inhib. hit(s) with Target = 'Vasopressin V1b receptor'
TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301669(US10131692, Compound 1)
Affinity DataEC50:  1.41E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301670(US10131692, Compound 2)
Affinity DataEC50:  8.07E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301671(US10131692, Compound 3)
Affinity DataEC50:  1.72E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301672(US10131692, Compound 4)
Affinity DataEC50:  2.49E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301673(US10131692, Compound 5)
Affinity DataEC50:  2.14E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301674(US10131692, Compound 6)
Affinity DataEC50:  5.76E+4nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301675(US10131692, Compound 7)
Affinity DataEC50:  1.42E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301676(US10131692, Compound 8)
Affinity DataEC50:  1.76E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301677(US10131692, Compound 9)
Affinity DataEC50: >1.00E+7nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301678(US10131692, Compound 10)
Affinity DataEC50:  1.05E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301679(US10131692, Compound 11)
Affinity DataEC50:  4.80E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301680(US10131692, Compound 12)
Affinity DataEC50:  3.22E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301681(US10131692, Compound 13)
Affinity DataEC50:  1.50E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301682(US10131692, Compound 14)
Affinity DataEC50:  1.88E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301683(US10131692, Compound 15)
Affinity DataEC50:  5.77E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301684(US10131692, Compound 27 | US10131692, Compound 16)
Affinity DataEC50:  4.81E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301685(US10131692, Compound 17)
Affinity DataEC50: >1.00E+7nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301686(US10131692, Compound 18)
Affinity DataEC50: >1.00E+7nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301687(US10131692, Compound 19)
Affinity DataEC50: >1.00E+7nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301688(US10131692, Compound 20)
Affinity DataEC50:  3.51E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301689(US10131692, Compound 21)
Affinity DataEC50:  5.36E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301690(US10131692, Compound 22)
Affinity DataEC50:  3.83E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301691(US10131692, Compound 23)
Affinity DataEC50:  5.18E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301692(US10131692, Compound 24)
Affinity DataEC50:  2.23E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301693(US10131692, Compound 25)
Affinity DataEC50:  6.43E+4nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301694(US10131692, Compound 26)
Affinity DataEC50:  4.58E+4nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301684(US10131692, Compound 27 | US10131692, Compound 16)
Affinity DataEC50:  1.33E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301696(US10131692, Compound 28)
Affinity DataEC50: >1.00E+7nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301697(US10131692, Compound 29)
Affinity DataEC50: >1.00E+7nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301698(US10131692, Compound 30)
Affinity DataEC50:  1.23E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301699(US10131692, Compound 31)
Affinity DataEC50:  2.58E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301700(US10131692, Compound 32)
Affinity DataEC50:  1.50E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301701(US10131692, Compound 33)
Affinity DataEC50:  1.60E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301702(US10131692, Compound 34)
Affinity DataEC50:  4.02E+4nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301703(US10131692, Compound 35)
Affinity DataEC50:  1.22E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301704(US10131692, Compound 36)
Affinity DataEC50:  9.56E+4nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301705(US10131692, Compound 37)
Affinity DataEC50:  1.01E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301706(US10131692, Compound 38)
Affinity DataEC50:  1.50E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301707(US10131692, Compound 39)
Affinity DataEC50:  3.29E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301708(US10131692, Compound 40)
Affinity DataEC50:  1.41E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301709(US10131692, Compound 41)
Affinity DataEC50:  1.14E+5nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM50205308(CHEMBL1429 | (S)-1-((4R,7S,10S,13S,16S)-7-(2-amino...)
Affinity DataEC50:  6.59E+3nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM301711(US10131692, Compound 43 ([Val4]dDAVP))
Affinity DataEC50:  2.41E+4nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM35667([3H]Argipressin tannate | AVP | [3H]Arginine vasop...)
Affinity DataEC50:  5.40E+3nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
US Patent

TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM50271606(CHEMBL4127791)
Affinity DataEC50:  8.30E+3nMAssay Description:Agonist activity at human vasopressin V1b receptor expressed in CHO cells assessed as increase in intracellular calcium flux measured for 5 mins by F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2020
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  33nMAssay Description:Agonist activity at human vasopressin V1b receptor expressed in CHO cells assessed as increase in intracellular calcium flux measured for 5 mins by F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2020
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM50271608(CHEMBL4129142)
Affinity DataEC50:  2.97E+3nMAssay Description:Agonist activity at human vasopressin V1b receptor expressed in CHO cells assessed as increase in intracellular calcium flux measured for 5 mins by F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2020
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM50271609(CHEMBL4128839)
Affinity DataEC50:  2.22E+3nMAssay Description:Agonist activity at human vasopressin V1b receptor expressed in CHO cells assessed as increase in intracellular calcium flux measured for 5 mins by F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2020
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM50271607(CHEMBL4126100)
Affinity DataEC50:  9.26E+3nMAssay Description:Agonist activity at human vasopressin V1b receptor expressed in CHO cells assessed as increase in intracellular calcium flux measured for 5 mins by F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2020
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Ferring

US Patent
LigandPNGBDBM50044677(CHEBI:59204 | Carbetocin)
Affinity DataEC50:  2.70E+4nMAssay Description:Agonist activity at human V1b receptor expressed in HEK293FT cells assessed as stimulation of calcium release by Aequorin based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
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