Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 12637
TargetVasopressin V1b receptor(Human)
Hmnc Holding

US Patent
LigandPNGBDBM50299343(SSR149415 | (2S,4R)-1-[5-Chloro-1-[(2,4-dimethoxyp...)
Affinity DataIC50: 1.5nMAssay Description:Test compounds were tested for binding to the V1b human vasopressin receptor using a human V1b (agonist radioligand) Receptor Binding Assay, with the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2025
Entry Details
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TargetVasopressin V1b receptor(Human)
Hmnc Holding

US Patent
LigandPNGBDBM716486(US20250034117, Compound Example 2)
Affinity DataIC50: 1.90nMAssay Description:Test compounds were tested for binding to the V1b human vasopressin receptor using a human V1b (agonist radioligand) Receptor Binding Assay, with the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2025
Entry Details
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TargetVasopressin V1b receptor(Human)
Hmnc Holding

US Patent
LigandPNGBDBM717676(US20250034117, Example 3)
Affinity DataIC50: 2nMAssay Description:Test compounds were tested for binding to the V1b human vasopressin receptor using a human V1b (agonist radioligand) Receptor Binding Assay, with the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2025
Entry Details
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TargetVasopressin V1b receptor(Human)
Hmnc Holding

US Patent
LigandPNGBDBM717675(US20250034117, Example 1)
Affinity DataIC50: 2.30nMAssay Description:Test compounds were tested for binding to the V1b human vasopressin receptor using a human V1b (agonist radioligand) Receptor Binding Assay, with the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2025
Entry Details
Go to US Patent

TargetVasopressin V1b receptor(Human)
Hmnc Holding

US Patent
LigandPNGBDBM50299343(SSR149415 | (2S,4R)-1-[5-Chloro-1-[(2,4-dimethoxyp...)
Affinity DataKi:  0.740nMAssay Description:Test compounds were tested for binding to the V1b human vasopressin receptor using a human V1b (agonist radioligand) Receptor Binding Assay, with the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2025
Entry Details
Go to US Patent

TargetVasopressin V1b receptor(Human)
Hmnc Holding

US Patent
LigandPNGBDBM716486(US20250034117, Compound Example 2)
Affinity DataKi:  0.960nMAssay Description:Test compounds were tested for binding to the V1b human vasopressin receptor using a human V1b (agonist radioligand) Receptor Binding Assay, with the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2025
Entry Details
Go to US Patent

TargetVasopressin V1b receptor(Human)
Hmnc Holding

US Patent
LigandPNGBDBM717676(US20250034117, Example 3)
Affinity DataKi:  0.980nMAssay Description:Test compounds were tested for binding to the V1b human vasopressin receptor using a human V1b (agonist radioligand) Receptor Binding Assay, with the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2025
Entry Details
Go to US Patent

TargetVasopressin V1b receptor(Human)
Hmnc Holding

US Patent
LigandPNGBDBM717675(US20250034117, Example 1)
Affinity DataKi:  1.20nMAssay Description:Test compounds were tested for binding to the V1b human vasopressin receptor using a human V1b (agonist radioligand) Receptor Binding Assay, with the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2025
Entry Details
Go to US Patent