27 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
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A dimeric urea of the bisabolene sesquiterpene from the Okinawan marine sponge Axinyssa sp. inhibits protein tyrosine phosphatase 1B activity in Huh-7 human hepatoma cells.
Tohoku Pharmaceutical University
Isomeric methoxy analogs of nimesulide for development of brain cyclooxygense-2 (COX-2)-targeted imaging agents: Synthesis, in vitro COX-2-inhibitory potency, and cellular transport properties.
Tohoku Pharmaceutical University
Strongylophorines, new protein tyrosine phosphatase 1B inhibitors, from the marine sponge Strongylophora strongilata collected at Iriomote Island.
Tohoku Pharmaceutical University
Verruculides A and B, two new protein tyrosine phosphatase 1B inhibitors from an Indonesian ascidian-derived Penicillium verruculosum.
Tohoku Pharmaceutical University
Structures and Biological Evaluations of Agelasines Isolated from the Okinawan Marine Sponge Agelas nakamurai.
Tohoku Pharmaceutical University
Absolute structures and bioactivities of euryspongins and eurydiene obtained from the marine sponge Euryspongia sp. collected at Iriomote Island.
Tohoku Pharmaceutical University
Two new protein tyrosine phosphatase 1B inhibitors, hyattellactones A and B, from the Indonesian marine sponge Hyattella sp.
Tohoku Pharmaceutical University
Synthesis and biological evaluation ofa-1-C-4'-arylbutyl-L-arabinoiminofuranoses, a new class ofa-glucosidase inhibitors.
Tohoku Pharmaceutical University
Novel estrogen receptor (ER) modulators containing various hydrophobic bent-core structures.
Tohoku Pharmaceutical University
Total synthesis of burkholdacs A and B and 5,6,20-tri-epi-burkholdac A: HDAC inhibition and antiproliferative activity.
Tohoku Pharmaceutical University
Euryspongins A-C, three new unique sesquiterpenes from a marine sponge Euryspongia sp.
Tohoku Pharmaceutical University
Total synthesis of bicyclic depsipeptides spiruchostatins C and D and investigation of their histone deacetylase inhibitory and antiproliferative activities.
Tohoku Pharmaceutical University
Synthesis and receptor binding properties of chimeric peptides containing a mu-opioid receptor ligand and nociceptin/orphanin FQ receptor ligand Ac-RYYRIK-amide.
Tohoku Pharmaceutical University
The synthesis and biological evaluation of 1-C-alkyl-L-arabinoiminofuranoses, a novel class ofa-glucosidase inhibitors.
Tohoku Pharmaceutical University
Matrix metalloproteinase-2 inhibitors from Clinopodium chinense var. parviflorum.
Tohoku Pharmaceutical University
Promising core structure for nuclear receptor ligands: design and synthesis of novel estrogen receptor ligands based on diphenylamine skeleton.
Tohoku Pharmaceutical University
Design and synthesis of carborane-containing androgen receptor (AR) antagonist bearing a pyridine ring.
Tohoku Pharmaceutical University
Synthesis of both enantiomers of hydroxypipecolic acid derivatives equivalent to 5-azapyranuronic acids and evaluation of their inhibitory activities against glycosidases.
Tohoku Pharmaceutical University
Synthesis of all stereoisomers of 3-hydroxypipecolic acid and 3-hydroxy-4,5-dehydropipecolic acid and their evaluation as glycosidase inhibitors.
Tohoku Pharmaceutical University
Utility of boron clusters for drug design. Relation between estrogen receptor binding affinity and hydrophobicity of phenols bearing various types of carboranyl groups.
Tohoku Pharmaceutical University
Dermorphin tetrapeptide analogues with 2',6'-dimethylphenylalanine (Dmp) substituted for aromatic amino acids have high mu opioid receptor binding and biological activities.
Tohoku Pharmaceutical University
Dermorphin and deltorphin heptapeptide analogues: replacement of Phe residue by Dmp greatly improves opioid receptor affinity and selectivity.
Tohoku Pharmaceutical University
Structure-activity studies on nociceptin analogues: ORL1 receptor binding and biological activity of cyclic disulfide-containing analogues of nociceptin peptides.
Tohoku Pharmaceutical University
Enkephalin analogues with 2',6'-dimethylphenylalanine replacing phenylalanine in position 4.
Tohoku Pharmaceutical University
Symmetric 4,4'-(piperidin-4-ylidenemethylene)bisphenol derivatives as novel tunable estrogen receptor (ER) modulators.
Tohoku Pharmaceutical University
Structure-activity relationship study on benzoic acid part of diphenylamine-based retinoids.
Tohoku Pharmaceutical University
