15 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
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Design of fluorinated 5-HT(4)R antagonists: influence of the basicity and lipophilicity toward the 5-HT(4)R binding affinities.
University of Southampton
Development of rationally designed DNA N6 adenine methyltransferase inhibitors.
University of Southampton
Binding constants of neuraminidase inhibitors: An investigation of the linear interaction energy method.
University of Southampton
Enantioselective synthesis of tranylcypromine analogues as lysine demethylase (LSD1) inhibitors.
University of Southampton
Small molecule agonists of the orphan nuclear receptors steroidogenic factor-1 (SF-1, NR5A1) and liver receptor homologue-1 (LRH-1, NR5A2).
University of Southampton
Exploring 2-Sulfonylpyrimidine Warheads as Acrylamide Surrogates for Targeted Covalent Inhibition: A BTK Story.
University of Southampton
Biophysical Survey of Small-Molecule β-Catenin Inhibitors: A Cautionary Tale.
University of Southampton
Systematic Investigation of Lipophilicity Modulation by Aliphatic Fluorination Motifs.
University of Southampton
Disubstituted Bis-THF Moieties as New P2 Ligands in Nonpeptidal HIV-1 Protease Inhibitors.
University of Southampton
Total Synthesis of Xanthoangelol B and Its Various Fragments: Toward Inhibition of Virulence Factor Production of Staphylococcus aureus.
University of Southampton
A genetically selected cyclic peptide inhibitor of BCL6 homodimerization.
University of Southampton
Aminobenzothiazole derivatives stabilize the thermolabile p53 cancer mutant Y220C and show anticancer activity in p53-Y220C cell lines.
University of Southampton
