65 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
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Design, synthesis, and evaluation of (2S,4R)-Ketoconazole sulfonamide analogs as potential treatments for Metabolic Syndrome.
Temple University
N-(2-Alkyleneimino-3-phenylpropyl)acetamide Compounds and Their Use against Pain and Pruritus via Inhibition of TRPA1 Channels.
Temple University
PPAR Agonists, Compounds, Pharmaceutical Compositions, and Methods of Use Thereof.
Temple University
PEGylated Bis-Sulfonamide Carbonic Anhydrase Inhibitors Can Efficiently Control the Growth of Several Carbonic Anhydrase IX-Expressing Carcinomas.
Temple University
Structure-Based Design, Synthesis, and Biological Evaluation of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2 Inhibitors.
Temple University
4,6-Diarylaminothiazines as BACE1 Inhibitors and Their Use for the Reduction of Beta-Amyloid Production.
Temple University
Biphenyl-ethyl-pyrrolidine derivatives as histamine h3 receptor modulators for the treatment of cognitive disorders.
Temple University
Imidazo[2,1]thiazol-3-one Derivatives Useful as Diagnostic Agents for Alzheimer's Disease.
Temple University
N-[4-(1H-Pyrazolo[3,4-B]pyrazin-6yl)-phenyl]-sulonamides and Their Use As Pharmaceuticals.
Temple University
Selective Cyp11B1 Inhibitors for the Treatment of Cortisol Dependent Diseases.
Temple University
Design, synthesis, and biological evaluation of 1-(4-sulfamylphenyl)-3-trifluoromethyl-5-indolyl pyrazolines as cyclooxygenase-2 (COX-2) and lipoxygenase (LOX) inhibitors.
Temple University
Design, synthesis and evaluation of (E)-alpha-benzylthio chalcones as novel inhibitors of BCR-ABL kinase.
Temple University
Identification of a chromone-based retinoid containing a polyolefinic side chain via facile synthetic routes.
Temple University
Discovery and SAR of Novel Disubstituted Quinazolines as Dual PI3Kalpha/mTOR Inhibitors Targeting Breast Cancer.
Temple University
Novel compounds that reverse the disease phenotype in Type 2 Gaucher disease patient-derived cells.
Temple University
Tricyclic Inhibitors of β-Secretase and Their Methods of Use for the Treatment of Alzheimer's Disease.
Temple University
Bridged Piperidine Derivatives Useful as γ-Secretase Inhibitors for the Treatment of Alzheimer's Disease.
Temple University
Triazolo Pyridines Useful as Inhibitors of γ-Secretase and Their Methods of Use.
Temple University
Design, synthesis, and evaluation of N-(4-(4-phenyl piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamides as selective dopamine D
Temple University
Modulators of KEAP-1 Activity as Potential Therapies for the Treatment of Neurodegenerative Disorders.
Temple University
Azabicyclic Fused Pyrimidine Derivatives Useful for the Treatment of Alzheimer's Disease.
Temple University
Azabicyclic Fused Pyrimidine Derivatives Useful for the Treatment of Alzheimer's Disease.
Temple University
Allosteric Modulators of Nicotinic Acetylcholine Receptors Useful for the Treatment of Cognitive Impairment.
Temple University
Covalent Inhibitors of the TEC Family of Kinases and Their Methods of Use.
Temple University
Novel inhibitors of Staphylococcus aureus RnpA that synergize with mupirocin.
Temple University
Interrogating the Roles of Post-Translational Modifications of Non-Histone Proteins.
Temple University
Design and synthesis of functionalized piperazin-1yl-(E)-stilbenes as inhibitors of 17α-hydroxylase-C17,20-lyase (Cyp17).
Temple University
Isolation of Acacetin from Calea urticifolia with Inhibitory Properties against Human Monoamine Oxidase-A and -B.
Temple University
Design, synthesis and SAR of new-di-substituted pyridopyrimidines as ATP-competitive dual PI3Kα/mTOR inhibitors.
Temple University
A CLASS OF FUSED RING COMPOUNDS, AND PREPARATION AND USE THEREOF
Cspc Zhongqi Pharmaceutical Technology (Shijiazhuang)
Novel multi-targeted agents for Alzheimer's disease: Synthesis, biological evaluation, and molecular modeling of novel 2-[4-(4-substitutedpiperazin-1-yl)phenyl]benzimidazoles
Hacettepe University